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PROTAC NAMPT Degrader-1
PROTAC NAMPT Degrader-1
SKU:QM-0101410
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Quantity
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Product Details
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Description
PROTAC NAMPT Degrader-1 is a potent PROTAC targeting NAMPT with aDC50 value of 217 nM. PROTAC NAMPT Degrader-1 has anti-proliferative activity with an IC50 value of 0.12μM against A2780 cells. (Structure Note: PINK, NAMPT activator ; Blue, VHL ligand (HY-163440) ; Black, linker).
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Molecular Formula
C57H69N13O8S2
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Molecular Weight
1128.37
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Smiles
O=C(NCC1=CC=NC=C1)NC2=CC=C(C=C2)S(=O)(N3CCN(CC3)C(C4=CC=C(C=C4)/N=N/C5=C(N(N=C5C)CCCCC(N[C@@H](C(C)(C)C)C(N6[C@@H](C[C@H](C6)O)C(N[C@H](C7=CC=C(C=C7)C8=C(N=CS8)C)C)=O)=O)=O)C)=O)=O
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Target
NAMPT; PROTACs
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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PROTAC NAMPT Degrader-1
PROTAC NAMPT Degrader-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.