PSB-0963 [CAS 1213268-73-5]

PSB-0963 is a selective and competitive ecto-5'-nucleotidase (eN/CD73) inhibitor with a Ki of 150 nM for rat ecto-5'-nucleotidase. PSB-0963 shows high selectivity over other ectonucleotidases (NTPDases 1-3) and P2Y receptors. PSB-0963 can be used for the study of cancer[1].

[1213268-73-5]

C28H17N2NaO5S

516.5

O=C1C2=C(C(C3=C(NC4=CC5=CC6=C(C=CC=C6)C=C5C=C4)C=C(S(=O)(O[Na])=O)C(N)=C13)=O)C=CC=C2

CD73

Room temperature