Name: PU139 [CAS 158093-65-3]
Brand: QuantiMol
SKU: QM-0141274-01
Price: 107.13 GBP
Availability: InStock

Product Details

Description
PU139 is a potent pan-histone acetyltransferase (HAT) inhibitor. PU139 blocks the HATs Gcn5, p300/CBP-associated factor (PCAF), CREB (cAMP response element-binding) protein (CBP) and p300 with IC50s of 8.39, 9.74, 2.49 and 5.35 μM, respectively[1][2].
CAS Number
[158093-65-3]
Molecular Formula
C12H7FN2OS
Molecular Weight
246.26
Smiles
O=C1N(C2=CC=C(F)C=C2)SC3=NC=CC=C31
Target
Histone Acetyltransferase
Isoform
CBP/p300; GCN5/PCAF
Purity
99.51
Solubility
DMSO : 10 mg/mL (ultrasonic; warming; heat to 60°C)
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Shipping Conditions
Room Temperature

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Variant	Variant total	Quantity	Price	Variant total
1 mgQM-0141274-01	1 mgQM-0141274-01 £107.13/ea	£0.00	Quantity	£107.13/ea	£0.00

5 mgQM-0141274-02	5 mgQM-0141274-02 £238.32/ea	£0.00	Quantity	£238.32/ea	£0.00

10 mM - 1 mLQM-0141274-03	10 mM - 1 mLQM-0141274-03 £290.57/ea	£0.00	Quantity	£290.57/ea	£0.00

10 mgQM-0141274-04	10 mgQM-0141274-04 £376.83/ea	£0.00	Quantity	£376.83/ea	£0.00

25 mgQM-0141274-05	25 mgQM-0141274-05 £670.87/ea	£0.00	Quantity	£670.87/ea	£0.00

50 mgQM-0141274-06	50 mgQM-0141274-06 £916.29/ea	£0.00	Quantity	£916.29/ea	£0.00

100 mgQM-0141274-07	100 mgQM-0141274-07 £1,267.43/ea	£0.00	Quantity	£1,267.43/ea	£0.00

250 mgQM-0141274-08	250 mgQM-0141274-08 £1,882.22/ea	£0.00	Quantity	£1,882.22/ea	£0.00

500 mgQM-0141274-09	500 mgQM-0141274-09 £2,685.34/ea	£0.00	Quantity	£2,685.34/ea	£0.00

1 gQM-0141274-10	1 gQM-0141274-10 £3,753.32/ea	£0.00	Quantity	£3,753.32/ea	£0.00

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