Raloxifene 4'-glucuronide-d4 [CAS 1279033-52-1]
Raloxifene 4'-glucuronide-d4 [CAS 1279033-52-1]
SKU:QM-0110873
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Product Details
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Description
Raloxifene 4'-glucuronide-d4 is deuterated labeled Raloxifene 4'-glucuronide. Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene. Raloxifene 4'-glucuronide formation is mediated mostly by UGT1A10 and UGT1A8. Raloxifene 4'-glucuronide binds to estrogen receptor with an IC50 of 370 μM.[2]. Raloxifene is a selective estrogen receptor modulator. Raloxifene activates TGFβ3 promoter as a full agonist at nanomolar concentrations, and inhibits the estrogen response element-containing vitellogenin promoter expression[3].
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CAS Number
[1279033-52-1]
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Molecular Formula
C34H31D4NO10S
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Molecular Weight
653.73
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Smiles
O=C(C1=CC=C(C=C1)OC([2H])([2H])C([2H])([2H])N2CCCCC2)C3=C(C4=CC=C(C=C4)O[C@@H]5O[C@@H]([C@H]([C@@H]([C@H]5O)O)O)C(O)=O)SC6=CC(O)=CC=C63
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Target
Estrogen Receptor/ERR; Isotope-Labeled Compounds
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Raloxifene 4'-glucuronide-d4 [CAS 1279033-52-1]
Raloxifene 4'-glucuronide-d4 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.