Raxlaprazine etomoxil [CAS 3034857-88-7]

Raxlaprazine etomoxil is a small molecule compound with dopamine D2 and D3 receptor modulating activity, which has potential application value in research related to mental illnesses. Raxlaprazine etomoxil exhibits high affinity for human recombinant D2L receptors, with an inhibition constant (Ki) of 1.95 nM. Raxlaprazine etomoxil effectively inhibits forskolin-stimulated cAMP accumulation, with an half maximal effective concentration (EC50) of 3.72 nM in functional activity experiments[1].

[3034857-88-7]

C23H36Cl2N4O2

471.46

ClC1=C(C=CC=C1Cl)N2CCN(CC2)CC[C@H]3CC[C@@H](CC3)NC(N(C)COCC)=O

Dopamine Receptor

Room temperature