Revefenacin-d4

Revefenacin-d4 (TD-4208-d4) is deuterium labeled Revefenacin. Revefenacin (TD-4208; GSK1160724) is a potent mAChR antagonist; has a high affinity on M3 receptor with a Ki of 0.18 nM.

C35H39D4N5O4

601.77

O=C(NC1=CC=CC=C1C2=CC=CC=C2)OC3CCN(CC3)CCN(C)C(C4=C(C([2H])=C(C([2H])=C4[2H])CN5CCC(CC5)C(N)=O)[2H])=O

Isotope-Labeled Compounds

Room temperature