Revefenacin-d9

Revefenacin-d9 (TD-4208-d9) is deuterium labeled Revefenacin. Revefenacin (TD-4208; GSK1160724) is a potent mAChR antagonist; has a high affinity on M3 receptor with a Ki of 0.18 nM.

C35H34D9N5O4

606.8

O=C(OC1CCN(CCN(C(C2=CC=C(CN3C([2H])([2H])C([2H])([2H])C(C(N)=O)([2H])C([2H])([2H])C3([2H])[2H])C=C2)=O)C)CC1)NC4=CC=CC=C4C5=CC=CC=C5

Isotope-Labeled Compounds

Room temperature