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Rimegepant (sulfate hydrate) [CAS 1374024-48-2]
Rimegepant (sulfate hydrate) [CAS 1374024-48-2]
SKU:QM-0007627-01
£200.66 GBP
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Product Details
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Description
Rimegepant (BMS-927711) sulfate hydrate is a potent, orally active, selective and competitive calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki of 0.027 nM and an IC50 of 0.14 nM for hCGRP receptor. Rimegepant sulfate hydrate can be used for migraine research[1][2][3].
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CAS Number
[1374024-48-2]
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Molecular Formula
C28H28F2N6O3.1/2H2O4S.3/2H2O
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Molecular Weight
610.26
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Smiles
O=S(O)(O)=O.O=C1N(C2CCN(CC2)C(O[C@H]3C4=NC=CC=C4[C@H]([C@H](C5=C(C(F)=CC=C5)F)CC3)N)=O)C6=CC=CN=C6N1.O.[0.5].[1.5]
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Target
CGRP Receptor
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Purity
99.48
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Solubility
DMSO : 7 mg/mL (ultrasonic)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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Rimegepant (sulfate hydrate) [CAS 1374024-48-2]
Rimegepant (sulfate hydrate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.