Risperidone-d6 [CAS 1225444-65-4]

Risperidone-d6 (R 64 766-d6) is the deuterium labeled Risperidone. Risperidone is a serotonin 5-HT2 receptor blocker, P-Glycoprotein inhibitor and potent dopamine D2 receptor antagonist, with Kis of 4.8, 5.9 nM for 5-HT2A and dopamine D2 receptor, respectively[1][2].

[1225444-65-4]

C23H21D6FN4O2

416.52

[2H]C([2H])(C1=C(C(N2CCCC([2H])(C2=N1)[2H])=O)CCN3CCC(CC3)C4=NOC5=C(C(F)=CC=C45)[2H])[2H]

5-HT Receptor; Dopamine Receptor; P-glycoprotein

5-HT2 Receptor; D2 Receptor; α-1 microglobulin

10 mM in DMSO

Room temperature