Roluperidone [CAS 359625-79-9]

Roluperidone (CYR-101) is a novel cyclic amide derivative that has high equipotent affinities for 5-HT2A and sigma-2 receptors (Ki of 7.53 nM and 8.19 nM for 5-HT2A and sigma-2, respectively) .

[359625-79-9]

C22H23FN2O2

366.43

O=C1N(CC2CCN(CC(C3=CC=C(F)C=C3)=O)CC2)CC4=C1C=CC=C4

5-HT Receptor; Sigma Receptor

5-HT2 Receptor; α-1 microglobulin

99.86

DMSO : 33.33 mg/mL (ultrasonic)

-20°C, 3 years; 4°C, 2 years (Powder)

Room Temperature