Sampatrilat [CAS 129981-36-8]
Sampatrilat [CAS 129981-36-8]
SKU:QM-0140846-01
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Product Details
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Description
Sampatrilat (UK-81252) is a potent and orally active vasopeptidase inhibitor of ACE and neutral endopeptidase (NEP) . Sampatrilat inhibits C-domain ACE (Ki=13.8 nM) 12.4-fold more potent than that for the N-domain (Ki=171.9 nM) . Sampatrilat (UK-81252) can be used for the study of chronic heart failure and blood pressure regulation[1][2].
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CAS Number
[129981-36-8]
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Molecular Formula
C26H40N4O9S
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Molecular Weight
584.68
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Smiles
OC([C@H](CNC([C@@H](NS(C)(=O)=O)CCCCN)=O)CC1(CCCC1)C(N[C@H](C(O)=O)CC2=CC=C(O)C=C2)=O)=O
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Target
Angiotensin-converting Enzyme (ACE) ; Neprilysin
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Purity
99.22
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Solubility
DMSO : 100 mg/mL (ultrasonic)
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Storage Conditions
-20°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Blue Ice
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Hazard Statement
H302-H312-H332
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Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P330-P363-P501
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Sampatrilat [CAS 129981-36-8]
Sampatrilat is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.