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SB 218795 [CAS 174635-53-1]

SB 218795 [CAS 174635-53-1]

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QM-0112687-01

£212.81 GBP
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Product Details

  • Description

    SB 218795 is a potent and selective non-peptide NK3 receptor antagonist, with a Ki 13 nM for hNK3. SB 218795 shows about 90-fold and 7000-fold selectivity for hNK3 over hNK2 and hNK1, respectively. SB 218795 can inhibit NK3 receptor-mediated pupillary constriction of the rabbit[1][2].

  • CAS Number

    [174635-53-1]

  • Molecular Formula

    C25H20N2O3

  • Molecular Weight

    396.44

  • Smiles

    COC([C@@H](C1=CC=CC=C1)NC(C2=CC(C3=CC=CC=C3)=NC4=CC=CC=C24)=O)=O

  • Target

    Neurokinin Receptor

  • Isoform

    NK2R; NK3R

  • Concentration

    10mM

  • Purity

    99.86

  • Solubility

    DMSO : 250 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302-H315-H319

  • Precautions

    P264-P270-P280-P302+P352-P305+P351+P338-P330-P362+P364-P501
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Variant Variant total Quantity Price Variant total
5 mgQM-0112687-01
5 mgQM-0112687-01
£212.81/ea		 £0.00
£212.81/ea £0.00
10 mM - 1 mLQM-0112687-02
10 mM - 1 mLQM-0112687-02
£229.82/ea		 £0.00
£229.82/ea £0.00
10 mgQM-0112687-03
10 mgQM-0112687-03
£313.65/ea		 £0.00
£313.65/ea £0.00
25 mgQM-0112687-04
25 mgQM-0112687-04
£577.31/ea		 £0.00
£577.31/ea £0.00
50 mgQM-0112687-05
50 mgQM-0112687-05
£902.93/ea		 £0.00
£902.93/ea £0.00
100 mgQM-0112687-06
100 mgQM-0112687-06
£1,405.94/ea		 £0.00
£1,405.94/ea £0.00
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SB 218795 [CAS 174635-53-1]

SB 218795 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.