Seladelpar (Lysine dihydrate) [CAS 928821-40-3]
Seladelpar (Lysine dihydrate) [CAS 928821-40-3]
SKU:QM-0085158-01
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Product Details
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Description
Seladelpar (MBX-8025) Lysine dihydrate is the Lysine dihydrate salt form of Seladelpar. Seladelpar Lysine dihydrate is an orally active agonist for potent PPAR-δ, with EC50 of 2 nM. Seladelpar Lysine dihydrate shows more than 750-fold and 2500-fold selectivity over the PPARα and PPARγ receptors, respectively. Seladelpar Lysine dihydrate can be used for the study of primary biliary cholangitis. Seladelpar Lysine dihydrate normalizes hyperglycemia, hyperinsulinemia, glucose, serum lipids and cholesterol levels, ameliorates the nonalcoholic steatohepatitis in mouse model[1][2].
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CAS Number
[928821-40-3]
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Molecular Formula
C27H41F3N2O9S
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Molecular Weight
626.68
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Smiles
N[C@@H](CCCCN)C(O)=O.O=C(O)COC1=CC=C(SC[C@H](OCC)COC2=CC=C(C(F)(F)F)C=C2)C=C1C.O.O
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Target
PPAR
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Isoform
PPARδ
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Purity
98
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Storage Conditions
4°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Room Temperature
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Seladelpar (Lysine dihydrate) [CAS 928821-40-3]
Seladelpar (Lysine dihydrate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.