ST1936 (oxalate) [CAS 1782228-83-4]

ST1936 oxalate is a selective, nanomolar affinity 5-HT6 receptor agonist with Ki values of 13 nM, 168 nM and 245 nM for human 5-HT6, 5-HT7 and 5-HT2B receptors, respectively. ST1936 oxalate also shows moderate affinity (Ki of 300 nM) for human and rat α2 adrenergic receptor[1].

[1782228-83-4]

C15H19ClN2O4

326.78

CC(N1)=C(CCN(C)C)C2=C1C=CC(Cl)=C2.O=C(O)C(O)=O

5-HT Receptor; Adrenergic Receptor

5-HT2 Receptor;5-HT6 Receptor;5-HT7 Receptor; MUC2; MUC3; α adrenergic receptor; α-1 microglobulin

10 mM in DMSO

Room temperature