T2857W

T2857W is a mutant peptide that has inhibitory effect on KIX-MLL interaction (IC50=5.67 μM) . T2857W can be used for protein-protein interaction (PPI) and for the study of diseases related to KIX-MLL interaction, such as leukemia, cancer, etc[1].

C68H101N15O19S

1464.68

O=C(N[C@@H](CO)C(N[C@@H](CC(O)=O)C(N[C@@H]([C@@H](C)CC)C(N[C@@H](CCSC)C(N[C@@H](CC(O)=O)C(N[C@@H](CC1=CC=CC=C1)C(N[C@@H](C(C)C)C(N[C@@H](CC(C)C)C(N[C@@H](CCCCN)C(N[C@@H](CC(N)=O)C(N[C@@H](CC2=CNC3=CC=CC=C23)C(O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)[C@H]4NCCC4

Histone Methyltransferase

Room temperature