Skip to product information
1 of 1

TEAD-IN-9

TEAD-IN-9

Size

SKU:QM-0092391

Price on request
Quantity

Request quote or documents

View full details
  • Description

    TEAD-IN-9 (compound 17) is a TEAD1 inhibitor with an IC50 of 0.29 μM. TEAD-IN-9 targets the palmitoyl pocket of TEAD, thereby effectively inhibiting the binding of YAP-TEAD and blocking the transcriptional function of YAP-TEAD[1].

  • Molecular Formula

    C23H23F3N3O3P

  • Molecular Weight

    477.42

  • Smiles

    O=P(C)(C)C1=CC=C(NCC2=CC=C(C(F)(F)F)C=C2)C(C3=NC(OC4COC4)=CC=N3)=C1

  • Target

    YAP

  • Isoform

    TEAD

  • Solubility

    10 mM in DMSO

  • Shipping Conditions

    Room temperature

Your cart
Variant Variant total Quantity Price Variant total
1 EachQM-0092391
1 EachQM-0092391
£0.00/ea
£0.00
£0.00/ea £0.00

TEAD-IN-9

TEAD-IN-9 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.