XY221

Name: XY221
Brand: QuantiMol
SKU: QM-0009264-01
Price: 2583.28 GBP
Availability: InStock

Size 5 mg 10 mg 25 mg 50 mg

SKU:QM-0009264-01

£2,583.28 GBP

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Product Details

Description
XY221 (Compound 16o) selectively inhibits BRD4 BD2, with an IC50 of 5.8 nM. XY221 demonstrates high pan-BD2 selectivity (667-fold over BRD4 BD1) and BRD4 BD2 domain selectivity (9−32-fold over BRD2/3/T BD2) . XY221 induce Apoptosis in MV4-11 cells and shows anticancer activity [1].
Molecular Formula
C32H34FN3O5
Molecular Weight
559.63
Smiles
O=C1C2=C(OC(C3=C(COC)N=C(CC)N3)=C2)C(C4=CC(C(C)(O)C)=CC=C4OC5=C(C)C=C(F)C=C5C)=CN1C
Target
AMPK; Apoptosis; Bcl-2 Family; c-Myc; Epigenetic Reader Domain; PAK
Isoform
BRD3; BRD4
Shipping Conditions
Room temperature

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Variant	Variant total	Quantity	Price	Variant total
5 mgQM-0009264-01	5 mgQM-0009264-01 £2,583.28/ea	£0.00	Quantity	£2,583.28/ea	£0.00

10 mgQM-0009264-02	10 mgQM-0009264-02 £3,849.30/ea	£0.00	Quantity	£3,849.30/ea	£0.00

25 mgQM-0009264-03	25 mgQM-0009264-03 £6,889.23/ea	£0.00	Quantity	£6,889.23/ea	£0.00

50 mgQM-0009264-04	50 mgQM-0009264-04 £10,992.29/ea	£0.00	Quantity	£10,992.29/ea	£0.00

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XY221 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.