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Y06137 [CAS 2226534-49-0]

Y06137 [CAS 2226534-49-0]

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QM-0137103-01

£250.47 GBP
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Product Details

  • Description

    Y06137 is a potent and selective BET inhibitor for treatment of castration-resistant prostate cancer (CRPC) . Y06137 binds to the BRD4 (1) bromodomain with a Kd of 81 nM[1].

  • CAS Number

    [2226534-49-0]

  • Molecular Formula

    C27H32N4O2

  • Molecular Weight

    444.57

  • Smiles

    CC1=NOC(C1=C2)=CC=C2C3=NC(C=C4)=C(N3CC5CCCCC5)C=C4N6CCOC[C@@H]6C

  • Target

    Epigenetic Reader Domain

  • Isoform

    BRD4

  • Purity

    99.9

  • Solubility

    DMSO : 62.5 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature
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Variant Variant total Quantity Price Variant total
5 mgQM-0137103-01
5 mgQM-0137103-01
£250.47/ea		 £0.00
£250.47/ea £0.00
10 mM - 1 mLQM-0137103-02
10 mM - 1 mLQM-0137103-02
£271.13/ea		 £0.00
£271.13/ea £0.00
10 mgQM-0137103-03
10 mgQM-0137103-03
£376.83/ea		 £0.00
£376.83/ea £0.00
25 mgQM-0137103-04
25 mgQM-0137103-04
£652.64/ea		 £0.00
£652.64/ea £0.00
50 mgQM-0137103-05
50 mgQM-0137103-05
£902.93/ea		 £0.00
£902.93/ea £0.00
100 mgQM-0137103-06
100 mgQM-0137103-06
£1,261.36/ea		 £0.00
£1,261.36/ea £0.00
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Y06137 [CAS 2226534-49-0]

Y06137 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.