Zanapezil (fumarate) [CAS 263248-42-6]
Zanapezil (fumarate) [CAS 263248-42-6]
SKU:QM-0074079
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Product Details
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Description
Zanapezil (TAK-147) fumarate is a potent, reversible and selective acetylcholine esterase (AChE) inhibitor. Zanapezil fumarate shows a potent and reversible inhibition of AChE activity in homogenates of the rat cerebral cortex (IC50=51.2 nM) . Zanapezil fumarate shows a moderate inhibition of muscarinic M1 and M2 receptor binding with Ki values of 234 and 340 nM, respectively. Zanapezil fumarate can be used for the research of early stages of Alzheimer's disease (AD) [1].
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CAS Number
[263248-42-6]
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Molecular Formula
C25H32N2O.xC4H4O4
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Smiles
OC(/C=C/C(O)=O)=O.O=C(C1=CC=C(CCCCN2)C2=C1)CCC3CCN(CC3)CC4=CC=CC=C4.[x]
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Target
Cholinesterase (ChE)
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Isoform
AChE
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Purity
99.63
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Solubility
10 mM in DMSO
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Storage Conditions
4°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Room Temperature
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Zanapezil (fumarate) [CAS 263248-42-6]
Zanapezil (fumarate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.