Name: Zeteletinib [CAS 2216753-97-6]
Brand: QuantiMol
SKU: QM-0146774-01
Price: 928.45 GBP
Availability: InStock

Product Details

Description
Zeteletinib (BOS-172738; DS-5010) is an orally active, selective RET kinase inhibitor with nanomolar potency against RET and >300-fold selectivity against VEGFR2. Zeteletinib shows exquisite potency for the wild type RET, RETV804M/L gatekeeper mutants, and the most common oncogenic RET mutation M918T. Zeteletinib has potent antitumor activity[1][2][3].
CAS Number
[2216753-97-6]
Molecular Formula
C25H23F3N4O4
Molecular Weight
500.47
Smiles
O=C(CC1=CC=C(C2=CN=C3C=C(C(OC)=CC3=C2)OC)N=C1)NC4=CC(C(C)(C(F)(F)F)C)=NO4
Target
PDGFR; RET
Isoform
PDGFR
Purity
98.31
Solubility
DMSO : 100 mg/mL (ultrasonic)
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Shipping Conditions
Room Temperature

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Variant	Variant total	Quantity	Price	Variant total
5 mgQM-0146774-01	5 mgQM-0146774-01 £928.45/ea	£0.00	Quantity	£928.45/ea	£0.00

10 mM - 1 mLQM-0146774-02	10 mM - 1 mLQM-0146774-02 £1,018.36/ea	£0.00	Quantity	£1,018.36/ea	£0.00

10 mgQM-0146774-03	10 mgQM-0146774-03 £1,430.24/ea	£0.00	Quantity	£1,430.24/ea	£0.00

25 mgQM-0146774-04	25 mgQM-0146774-04 £2,873.66/ea	£0.00	Quantity	£2,873.66/ea	£0.00

50 mgQM-0146774-05	50 mgQM-0146774-05 £4,568.59/ea	£0.00	Quantity	£4,568.59/ea	£0.00

100 mgQM-0146774-06	100 mgQM-0146774-06 £7,330.28/ea	£0.00	Quantity	£7,330.28/ea	£0.00

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Zeteletinib [CAS 2216753-97-6]

Zeteletinib is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.