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Aldumastat [CAS 1957278-93-1]

Aldumastat [CAS 1957278-93-1]

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SKU:QM-0145957-01

£301.50 GBP
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  • Description

    Aldumastat (GLPG1972; S201086) is a potent, seletive and orally active ADAMTS-5 (IC50=19 nM) inhibitor, and has 8-fold seletivity over ADAMTS-4 (IC50=156 nM) . Aldumastat has anticatabolic activity and is used for osteoarthritis research[1].

  • CAS Number

    [1957278-93-1]

  • Molecular Formula

    C20H24F2N4O3

  • Molecular Weight

    406.43

  • Smiles

    O=C(N(CCN1C2=CC(F)=CC(F)=C2)C[C@@H]1C)CC[C@](NC3=O)(C4CC4)C(N3)=O

  • Target

    ADAMTS

  • Isoform

    MMP-14; MMP-2

  • Purity

    99.36

  • Solubility

    DMSO : 100 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H315, H319, H335

  • Precautions

    H315, H319, H335

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Variant Variant total Quantity Price Variant total
1 mgQM-0145957-01
1 mgQM-0145957-01
£301.50/ea
£0.00
£301.50/ea £0.00
5 mgQM-0145957-02
5 mgQM-0145957-02
£678.15/ea
£0.00
£678.15/ea £0.00
10 mM - 1 mLQM-0145957-03
10 mM - 1 mLQM-0145957-03
£740.12/ea
£0.00
£740.12/ea £0.00
10 mgQM-0145957-04
10 mgQM-0145957-04
£1,116.77/ea
£0.00
£1,116.77/ea £0.00
25 mgQM-0145957-05
25 mgQM-0145957-05
£2,309.90/ea
£0.00
£2,309.90/ea £0.00
50 mgQM-0145957-06
50 mgQM-0145957-06
£3,815.28/ea
£0.00
£3,815.28/ea £0.00
100 mgQM-0145957-07
100 mgQM-0145957-07
£5,823.68/ea
£0.00
£5,823.68/ea £0.00

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Aldumastat [CAS 1957278-93-1]

Aldumastat is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.