1 1

Apitolisib [CAS 1032754-93-0]

Apitolisib [CAS 1032754-93-0]

Size

QM-0144018-01

£115.00 GBP
Sale Sold out

Request quote or documents

View full details

Product Details

  • Description

    Apitolisib (GDC-0980; GNE 390; RG 7422) is a selective, potent, orally bioavailable Class I PI3 kinase and mTOR kinase (TORC1/2) inhibitor with IC50s of 5 nM/27 nM/7 nM/14 nM for PI3Kα/PI3Kβ/PI3Kδ/PI3Kγ, and with a Ki of 17 nM for mTOR.

  • CAS Number

    [1032754-93-0]

  • Molecular Formula

    C23H30N8O3S

  • Molecular Weight

    498.6

  • Smiles

    C[C@@H](C(N1CCN(CC1)CC2=C(C3=NC(C4=CN=C(N=C4)N)=NC(N5CCOCC5)=C3S2)C)=O)O

  • Target

    Apoptosis; mTOR; PI3K

  • Isoform

    MTOR; mTORC1; mTORC2; PI3Kα; PI3Kβ; PI3Kγ; PI3Kδ

  • Concentration

    10mM

  • Purity

    99.29

  • Solubility

    DMSO : 14.29 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302, H315, H319, H335

  • Precautions

    H302, H315, H319, H335
Learn more
Variant Variant total Quantity Price Variant total
5 mgQM-0144018-01
5 mgQM-0144018-01
£115.00/ea		 £0.00
£115.00/ea £0.00
10 mM - 1 mLQM-0144018-02
10 mM - 1 mLQM-0144018-02
£124.00/ea		 £0.00
£124.00/ea £0.00
10 mgQM-0144018-03
10 mgQM-0144018-03
£188.51/ea		 £0.00
£188.51/ea £0.00
50 mgQM-0144018-04
50 mgQM-0144018-04
£450.95/ea		 £0.00
£450.95/ea £0.00
100 mgQM-0144018-05
100 mgQM-0144018-05
£726.75/ea		 £0.00
£726.75/ea £0.00
View cart
0

Total items

£0.00

Product subtotal

Taxes, discounts and shipping calculated at checkout.
View cart

Related Products

Other industry favorites

Apitolisib [CAS 1032754-93-0]

Apitolisib is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.