CARM1-IN-1 (hydrochloride) [CAS 2070018-31-2]
CARM1-IN-1 (hydrochloride) [CAS 2070018-31-2]
SKU:QM-0142208-01
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Product Details
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Description
CARM1-IN-1 (compound 7g) hydrochloride is a highly potent and selective inhibitor of CARM1 (IC50=8.6 μM, CARM1/PABP1), with low inhibitory activity against PRMT1 and SET7 (IC50 >667 μM) . CARM1-IN-1 hydrochloride inhibits the methylation activity of CARM1 and the methylation levels of different substrates, such as PABP1, CA150, SmB, and H3. CARM1-IN-1 hydrochloride also inhibits the promoter activity of prostate-specific antigen (PSA) without significant cytotoxicity[1].
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CAS Number
[2070018-31-2]
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Molecular Formula
C26H22Br2ClNO3
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Molecular Weight
591.72
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Smiles
[H]Cl.O=C1/C(CN(CC2=CC=CC=C2)C/C1=C\C3=CC=C(O)C(Br)=C3)=C/C4=CC=C(O)C(Br)=C4
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Target
Histone Methyltransferase
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Isoform
PRMT4
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Purity
95.13
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Solubility
DMSO : 250 mg/mL (ultrasonic)
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Storage Conditions
4°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Room Temperature
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CARM1-IN-1 (hydrochloride) [CAS 2070018-31-2]
CARM1-IN-1 (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.