CEP-28122 (mesylate salt) [CAS 2070009-30-0]
CEP-28122 (mesylate salt) [CAS 2070009-30-0]
SKU:QM-0154845-01
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Product Details
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Description
CEP-28122 mesylate salt, a diaminopyrimidine derivative, is a potent, selective, and orally bioavailable ALK inhibitor, with an IC50 value of 1.9 nM for recombinant ALK kinase activity. CEP-28122 has antitumor activity in experimental models of ALK-positive human cancers. CEP-28122 mesylate salt has good pharmacodynamic and pharmacokinetic activity[1].
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CAS Number
[2070009-30-0]
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Molecular Formula
C29H39ClN6O6S
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Molecular Weight
635.17
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Smiles
O=C([C@H]1[C@](C2)([H])C=C[C@]2([H])[C@H]1NC3=NC(NC4=CC=C5C(CC[C@@H](N6CCOCC6)CC5)=C4OC)=NC=C3Cl)N.O=S(C)(O)=O
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Target
Anaplastic lymphoma kinase (ALK)
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Concentration
10mM
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Purity
99.92
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Solubility
DMSO : 6.4 mg/mL (ultrasonic; warming)
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Storage Conditions
4°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Room Temperature
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CEP-28122 (mesylate salt) [CAS 2070009-30-0]
CEP-28122 (mesylate salt) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.