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CGP 12177 (hydrochloride) [CAS 64208-32-8]

CGP 12177 (hydrochloride) [CAS 64208-32-8]

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SKU:QM-0081206-01

£249.26 GBP
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  • Description

    CGP 12177 ((±) -CGP 12177) hydrochloride is a β-Adrenergic receptor (β-AR) ligand. CGP 12177 hydrochloride is a β3-AR (Ki = 88 nM) agonist with β1/β2-AR (Ki = 0.9 nM for β1; Ki = 4 nM for β2) antagonist action. CGP 12177 hydrochloride exhibits partial agonist properties for α1-AR in rat pulmonary artery. CGP 12177 hydrochloride regulates the expression of ucp and leptin genes in NMRI mice adipose tissues. CGP 12177 hydrochloride can be used for cardiovascular and metabolic disease research[1][2][3][4].

  • CAS Number

    [64208-32-8]

  • Molecular Formula

    C14H22ClN3O3

  • Molecular Weight

    315.8

  • Smiles

    O=C1NC2=C(OCC(O)CNC(C)(C)C)C=CC=C2N1.Cl

  • Target

    Adrenergic Receptor

  • Isoform

    α adrenergic receptor; β adrenergic receptor

  • Purity

    99.69

  • Solubility

    DMSO : 10 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C (Powder, sealed storage, away from moisture)

  • Shipping Conditions

    Blue Ice

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Variant Variant total Quantity Price Variant total
5 mgQM-0081206-01
5 mgQM-0081206-01
£249.26/ea
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10 mgQM-0081206-02
10 mgQM-0081206-02
£368.33/ea
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CGP 12177 (hydrochloride) [CAS 64208-32-8]

CGP 12177 (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.