Dagrocorat (hydrochloride) [CAS 1044535-61-6]
Dagrocorat (hydrochloride) [CAS 1044535-61-6]
SKU:QM-0154051-01
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Product Details
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Description
Dagrocorat (PF-00251802) hydrochloride is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat hydrochloride is also a time-dependent reversible inhibitor of CYP3A (IC50=1.3 μM in human liver microsomes) and CYP2D6 (Ki=0.57 μM in human liver microsomes) . Dagrocorat hydrochloride can be used for the research of rheumatoid arthritis[1].
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CAS Number
[1044535-61-6]
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Molecular Formula
C29H30ClF3N2O2
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Molecular Weight
531.01
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Smiles
O[C@@]1(C(F)(F)F)C[C@]2([H])[C@](C3=CC=C(C(NC(C=CC=N4)=C4C)=O)C=C3CC2)(CC1)CC5=CC=CC=C5.[H]Cl
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Target
Cytochrome P450; Glucocorticoid Receptor
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Isoform
CYP2; CYP3
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Purity
99.85
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Solubility
DMSO : 100 mg/mL (ultrasonic; warming; heat to 60°C)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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Dagrocorat (hydrochloride) [CAS 1044535-61-6]
Dagrocorat (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.