Dapitant [CAS 153438-49-4]
Dapitant [CAS 153438-49-4]
SKU:QM-0076091
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Product Details
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Description
Dapitant (RPR 100893) is a non-peptide Substance P antagonist with high affinity for the human NK1 receptor. It belongs to the 7,7,4-trimethylperhydroisoindole class of compounds. Dapitant inhibits the binding of Substance P to NK1 receptors, thereby blocking its neurokinin-mediated effects. This novel antagonist represents a potential therapeutic option for conditions involving Substance P, such as neurogenic inflammation and pain modulation[1].
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CAS Number
[153438-49-4]
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Molecular Formula
C37H39NO4
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Molecular Weight
561.71
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Smiles
COC1=CC=CC=C1[C@]2(O)CCC(C3=CC=CC=C3)(C4=CC=CC=C4)[C@]5([H])[C@@]2([H])CN(C([C@@H](C)C6=C(OC)C=CC=C6)=O)C5
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Target
Neurokinin Receptor
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Shipping Conditions
Room temperature
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Dapitant [CAS 153438-49-4]
Dapitant is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.