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Darbufelone (mesylate) [CAS 139340-56-0]
Darbufelone (mesylate) [CAS 139340-56-0]
SKU:QM-0081260-01
£212.81 GBP
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Product Details
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Description
Darbufelone mesylate (CI-1004 mesylate) is a dual inhibitor of cellular PGF2α and LTB4 production. Darbufelone potently inhibits PGHS-2 (IC50 = 0.19 μM) but is much less potent with PGHS-1 (IC50= 20 μM) .
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CAS Number
[139340-56-0]
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Molecular Formula
C19H28N2O5S2
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Molecular Weight
428.57
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Smiles
O=C1N=C(N)S/C1=C\C2=CC(C(C)(C)C)=C(O)C(C(C)(C)C)=C2.CS(=O)(O)=O
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Target
Leukotriene Receptor; Prostaglandin Receptor
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Isoform
FP; LTB4
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Concentration
10mM
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Purity
99.65
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Solubility
DMSO : 110 mg/mL (ultrasonic) |H2O : < 0.1 mg/mL (ultrasonic; warming; heat to 60°C)
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Storage Conditions
4°C (Powder, sealed storage, away from moisture and light)
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Shipping Conditions
Room Temperature
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Darbufelone (mesylate) [CAS 139340-56-0]
Darbufelone (mesylate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.