DOTA.SA.FAPi (TFA)
DOTA.SA.FAPi (TFA)
SKU:QM-0161289-01
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Product Details
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Description
DOTA.SA.FAPi TFA inhibits fibroblast activation protein (FAP) with an IC50 of 0.9 nM. DOTA.SA.FAPi TFA targets protease PREP with an IC50 of 5.4 μM. DOTA.SA.FAPi TFA can be used a PET tracer, when labeled with 68Ga, and used for research about cancer[1]. DOTA.SA.FAPi (TFA) can be used for the synthesis/research of Radionuclide-Drug Conjugates (RDCs) .
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Molecular Formula
C45H56F5N11O14
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Molecular Weight
1069.98
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Smiles
O=C(O)CN1CCN(CC(O)=O)CCN(CC(O)=O)CCN(CC(NCCNC(C2=O)=C(NCCCCOC3=CC(C(C(NCC(N4[C@H](C#N)CC(F)(F)C4)=O)=O)=CC=N5)=C5C=C3)C2=O)=O)CC1.OC(C(F)(F)F)=O
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Target
FAP; Prolyl Endopeptidase (PREP) ; Radionuclide-Drug Conjugates (RDCs)
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Isoform
RDC Peptide
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Purity
99.26
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Solubility
H2O : ≥ 50 mg/mL
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Storage Conditions
-20°C (Powder, sealed storage, away from moisture and light)
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Shipping Conditions
Blue Ice
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DOTA.SA.FAPi (TFA)
DOTA.SA.FAPi (TFA) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.