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EPAC 5376753 [CAS 302826-61-5]
EPAC 5376753 [CAS 302826-61-5]
SKU:QM-0137068-01
£210.38 GBP
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Product Details
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Description
EPAC 5376753, a 2-Thiobarbituric acid derivative, is a selective and allosteric Epac inhibitor. EPAC 5376753 inhibits Epac1 with an IC50 of 4 µM in Swiss 3T3 cells. EPAC 5376753 does not inhibit PKA and adenylyl cyclases[1].
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CAS Number
[302826-61-5]
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Molecular Formula
C15H8Cl2N2O3S
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Molecular Weight
367.21
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Smiles
O=C(/C(C(N1)=O)=C/C2=CC=C(C3=CC=C(Cl)C=C3Cl)O2)NC1=S
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Target
Ras
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Purity
98.1
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Solubility
10 mM in DMSO
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Storage Conditions
4°C (Powder, protect from light)
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Shipping Conditions
Room Temperature
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EPAC 5376753 [CAS 302826-61-5]
EPAC 5376753 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.