Ezatiostat (hydrochloride) [CAS 286942-97-0]
Ezatiostat (hydrochloride) [CAS 286942-97-0]
SKU:QM-0000475
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Product Details
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Description
Ezatiostat hydrochloride (TER199; TLK199 hydrochloride) is a tripeptide analog of glutathione and is a selective and orally active glutathione S-transferase P1-1 (GSTP1) inhibitor. Ezatiostat hydrochloride leads to JNK activation by inhibiting GSTP1. Ezatiostat hydrochloride stimulates both lymphocyte production and bone marrow progenitor proliferation. Ezatiostat hydrochloride has the potential for myelodysplastic syndrome (MDS) treatment[1][2].
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CAS Number
[286942-97-0]
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Molecular Formula
C27H36ClN3O6S
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Molecular Weight
566.11
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Smiles
O=C(OCC)[C@@H](C1=CC=CC=C1)NC([C@@H](NC(CC[C@H](N)C(OCC)=O)=O)CSCC2=CC=CC=C2)=O.Cl
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Target
Apoptosis; Glutathione S-transferase
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Ezatiostat (hydrochloride) [CAS 286942-97-0]
Ezatiostat (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.