Skip to product information
1 of 1

F-14512 (hydrochloride) [CAS 866874-39-7]

F-14512 (hydrochloride) [CAS 866874-39-7]

Size

SKU:QM-0002986

Price on request
Quantity

Request quote or documents

View full details
  • Description

    F-14512 hydrochloride is an anticancer agent that utilizes the polyamine transport system (PTS) to selectively deliver polyamine-containing drugs to cancer cells. F-14512 hydrochloride enhances the affinity of polyamines for DNA, thereby inhibiting topoisomerase II and achieving selective cellular uptake. F-14512 hydrochloride exhibits significant cytotoxicity against cells with high PTS activity and induces DNA damage. F-14512 hydrochloride demonstrates potent antitumor activity in the MX1 breast tumor xenograft model. F-14512 hydrochloride could be used to study breast cancer[1].

  • CAS Number

    [866874-39-7]

  • Molecular Formula

    C33H51Cl4N5O8

  • Molecular Weight

    787.6

  • Smiles

    O=C1[C@]2([H])[C@H](C3=CC(OC)=C(C(OC)=C3)O)C4=CC(OCO5)=C5C=C4[C@H]([C@@]2([H])CO1)NC(CNCCCNCCCCNCCCN)=O.Cl.Cl.Cl.Cl

  • Target

    DNA/RNA Synthesis; Topoisomerase

  • Shipping Conditions

    Room temperature

Your cart
Variant Variant total Quantity Price Variant total
1 EachQM-0002986
1 EachQM-0002986
£0.00/ea
£0.00
£0.00/ea £0.00

F-14512 (hydrochloride) [CAS 866874-39-7]

F-14512 (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.