GR127935 (hydrochloride) [CAS 148642-42-6]
GR127935 (hydrochloride) [CAS 148642-42-6]
SKU:QM-0056952-01
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Product Details
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Description
GR127935 hydrochloride is a potent and orally active 5-HT1D and 5-HT1B receptor antagonist with pKis of 8.5 for both isoforms. GR127935 hydrochloride has 100-fold selectivity for 5-HT1B/1D receptors over 5-HT1A, 5-HT2A, and 5-HT2C receptors. GR127935 hydrochloride can be used in neurological disease research[1][2].
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CAS Number
[148642-42-6]
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Molecular Formula
C29H32ClN5O3
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Molecular Weight
534.05
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Smiles
O=C(C1=CC=C(C2=CC=C(C3=NOC(C)=N3)C=C2C)C=C1)NC4=CC=C(OC)C(N5CCN(C)CC5)=C4.[H]Cl
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Target
5-HT Receptor
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Isoform
5-HT1 Receptor;5-HT2 Receptor; mLAG-3
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Purity
99.38
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Solubility
DMSO : 83.33 mg/mL (ultrasonic)
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Storage Conditions
-20°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Blue Ice
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Hazard Statement
H315, H319
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Precautions
H315, H319
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GR127935 (hydrochloride) [CAS 148642-42-6]
GR127935 (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.