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Grapiprant [CAS 415903-37-6]

Grapiprant [CAS 415903-37-6]

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QM-0154145-01

£129.63 GBP
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Product Details

  • Description

    Grapiprant (CJ-023423) is a selective EP4 receptor antagonist whose physiological ligand is prostaglandin E2 (PGE2) . Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor with IC50 value of 35 nM and Ki value of 24 nM. Grapiprant has the potential for osteoarthritic pain and inflammation treatment[1][2][3] .

  • CAS Number

    [415903-37-6]

  • Molecular Formula

    C26H29N5O3S

  • Molecular Weight

    491.61

  • Smiles

    O=S(C1=CC=C(C)C=C1)(NC(NCCC2=CC=C(N3C(CC)=NC4=C3C=C(C)N=C4C)C=C2)=O)=O

  • Target

    Prostaglandin Receptor

  • Isoform

    EP

  • Purity

    99.57

  • Solubility

    DMSO : ≥ 50 mg/mL

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302

  • Precautions

    H302
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Variant Variant total Quantity Price Variant total
5 mgQM-0154145-01
5 mgQM-0154145-01
£129.63/ea		 £0.00
£129.63/ea £0.00
10 mM - 1 mLQM-0154145-02
10 mM - 1 mLQM-0154145-02
£139.75/ea		 £0.00
£139.75/ea £0.00
10 mgQM-0154145-03
10 mgQM-0154145-03
£238.32/ea		 £0.00
£238.32/ea £0.00
25 mgQM-0154145-04
25 mgQM-0154145-04
£363.47/ea		 £0.00
£363.47/ea £0.00
50 mgQM-0154145-05
50 mgQM-0154145-05
£614.98/ea		 £0.00
£614.98/ea £0.00
100 mgQM-0154145-06
100 mgQM-0154145-06
£953.96/ea		 £0.00
£953.96/ea £0.00
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Grapiprant [CAS 415903-37-6]

Grapiprant is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.