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Indole-2-carboxylic acid [CAS 1477-50-5]

Indole-2-carboxylic acid [CAS 1477-50-5]

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SKU:QM-0161552-01

£51.91 GBP
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  • Description

    Indole-2-carboxylic acid (I2CA) is a competitive antagonist of the glycine site of the NMDA receptor (Ki=15 μM, 5-fluoro-I2CA) and an inhibitor of HIV-1 integrase. Indole-2-carboxylic acid is selective for the glycine site of the NMDA receptor and blocks the enhancement of NMDA receptor by competitively inhibiting the binding of glycine to the NMDA receptor. Indole-2-carboxylic acid can also inhibit the strand transfer activity of HIV-1 integrase by chelating Mg2+ at the active site of integrase and interacting with the hydrophobic cavity. Indole-2-carboxylic acid can be used in the study of neurological diseases (such as stroke, epilepsy) and HIV-1 infection[1][2].

  • CAS Number

    [1477-50-5]

  • Molecular Formula

    C9H7NO2

  • Molecular Weight

    161.16

  • Smiles

    O=C(C(N1)=CC2=C1C=CC=C2)O

  • Target

    HIV; HIV Integrase; iGluR

  • Isoform

    Human Endogenous Metabolite; NMDA Receptor

  • Purity

    99.97

  • Solubility

    DMSO : 100 mg/mL (ultrasonic) |H2O : < 0.1 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302, H315, H319, H335

  • Precautions

    H302, H315, H319, H335

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5 gQM-0161552-01
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10 mM - 1 mLQM-0161552-02
10 mM - 1 mLQM-0161552-02
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10 gQM-0161552-03
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25 gQM-0161552-04
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50 gQM-0161552-05
50 gQM-0161552-05
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100 gQM-0161552-06
100 gQM-0161552-06
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Indole-2-carboxylic acid [CAS 1477-50-5]

Indole-2-carboxylic acid is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.