Lesogaberan (hydrochloride) [CAS 2925644-17-1]
Lesogaberan (hydrochloride) [CAS 2925644-17-1]
SKU:QM-0079515-01
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Product Details
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Description
Lesogaberan (AZD-3355) hydrochloride is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptor. The affinity (Kis) of Lesogaberan hydrochloride for rat GABAB and GABAA receptors, as measured by displacement of [3H]GABA binding in brain membranes: 5.1 nM and 1.4 μM, respectively. Lesogaberan hydrochloride inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action[1].
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CAS Number
[2925644-17-1]
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Molecular Formula
C3H10ClFNO2P
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Molecular Weight
177.54
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Smiles
O=P(C[C@H](F)CN)O.[H]Cl
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Target
GABA Receptor
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Purity
98
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Solubility
DMSO : 240 mg/mL (ultrasonic) |H2O : 100 mg/mL (ultrasonic)
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Storage Conditions
4°C (Powder, stored under nitrogen, away from moisture)
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Shipping Conditions
Room Temperature
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Lesogaberan (hydrochloride) [CAS 2925644-17-1]
Lesogaberan (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.