Lumateperone (tosylate) [CAS 1187020-80-9]
Lumateperone (tosylate) [CAS 1187020-80-9]
SKU:QM-0155492-01
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Product Details
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Description
Lumateperone (ITI-007) tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator. Lumateperone tosylate has anticancer activity and can also be used in studies of psychiatric disorders such as schizophrenia[1][2][3].
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CAS Number
[1187020-80-9]
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Molecular Formula
C31H36FN3O4S
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Molecular Weight
565.7
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Smiles
O=C(C1=CC=C(F)C=C1)CCCN2CC[C@@](N3CCN(C)C4=C3C5=CC=C4)([H])[C@@]5([H])C2.O=S(C6=CC=C(C)C=C6)(O)=O
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Target
5-HT Receptor; Dopamine Receptor
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Isoform
5-HT2 Receptor; D1 Receptor; D2 Receptor; α-1 microglobulin
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Purity
99.78
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Solubility
DMSO : 100 mg/mL (ultrasonic) |H2O : < 0.1 mg/mL (ultrasonic; warming; heat to 80°C)
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Storage Conditions
4°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Room Temperature
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Hazard Statement
H302, H315, H319, H335
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Precautions
H302, H315, H319, H335
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Lumateperone (tosylate) [CAS 1187020-80-9]
Lumateperone (tosylate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.