Opiranserin (hydrochloride) [CAS 1440796-75-7]
Opiranserin (hydrochloride) [CAS 1440796-75-7]
SKU:QM-0136381-01
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Product Details
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Description
Opiranserin (VVZ-149) hydrochloride, a non-opioid and non-NSAID analgesic candidate, is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. Opiranserin hydrochloride shows antagonistic activity on rP2X3 (IC50=0.87 μM) . Opiranserin hydrochloride is development as an injectable agent for the treatment of postoperative pain[1][2][3].
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CAS Number
[1440796-75-7]
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Molecular Formula
C21H35ClN2O5
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Molecular Weight
430.97
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Smiles
O=C(C1=CC(OC)=C(OCCCC)C(OC)=C1)NCC2(CCOCC2)N(C)C.[H]Cl
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Target
5-HT Receptor; GlyT; P2X Receptor
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Isoform
5-HT2 Receptor; GlyT2; P2X3 Receptor; α-1 microglobulin
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Concentration
10mM
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Purity
99.62
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Solubility
DMSO : 50 mg/mL (ultrasonic)
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Storage Conditions
4°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Room Temperature
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Opiranserin (hydrochloride) [CAS 1440796-75-7]
Opiranserin (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.