Pepstatin (Trifluoroacetate)
Pepstatin (Trifluoroacetate)
SKU:QM-0199403-01
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Product Details
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Description
Pepstatin (Pepstatin A) Trifluoroacetate is a specific, orally active aspartic protease inhibitor produced by actinomycetes, with IC50s of 4.5 nM, 6.2 nM, 150 nM, 290 nM, 520 nM and 260 nM for hemoglobin-pepsin, hemoglobin-proctase, casein-pepsin, casein-proctase, casein-acid protease and hemoglobin-acid protease, respectively. Pepstatin Trifluoroacetate also inhibits HIV protease[1][2].
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Molecular Formula
C36H64F3N5O11
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Molecular Weight
799.92
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Smiles
OC(C(F)(F)F)=O.CC(C[C@H](NC([C@@H](NC([C@@H](NC(CC(C)C)=O)C(C)C)=O)C(C)C)=O)[C@@H](O)CC(N[C@@H](C)C(N[C@@H](CC(C)C)[C@@H](O)CC(O)=O)=O)=O)C
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Target
Autophagy; HIV Protease
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Purity
99.13
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Solubility
DMSO : 25 mg/mL (ultrasonic)
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Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
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Shipping Conditions
Blue Ice
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Pepstatin (Trifluoroacetate)
Pepstatin (Trifluoroacetate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.