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PI3Kδ-IN-8 [CAS 2101518-75-4]
PI3Kδ-IN-8 [CAS 2101518-75-4]
SKU:QM-0062480
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Product Details
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Description
PI3Kδ-IN-8 is a potent, selective and orally active PI3Kδ inhibitor, with an IC50 of 3.3 nM. PI3Kδ-IN-8 shows selectivity for PI3Kδ over PI3Kα, PI3Kβ, and PI3Kγ (IC50=377.2, 241.6, 17.9 nM, respectively) . PI3Kδ-IN-8 has anti-tumor activity[1].
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CAS Number
[2101518-75-4]
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Molecular Formula
C28H21F2N7O
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Molecular Weight
509.51
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Smiles
N#CC1=C(N[C@H](C(C(C2=CC=C(F)C=C2)=C3C=CC(F)=CN43)=C(C5=CC=CC=C5)C4=O)C)N=C(N)N=C1N
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Target
PI3K
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Isoform
PI3Kα; PI3Kβ; PI3Kγ; PI3Kδ
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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PI3Kδ-IN-8 [CAS 2101518-75-4]
PI3Kδ-IN-8 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.