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PKRA83 (hydrochloride)
PKRA83 (hydrochloride)
SKU:QM-0007150
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Product Details
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Description
PKRA83 (PKRA7) hydrochloride is a potent, blood-brain-penetrating PK2 antagonist that competes for PK2 binding to its receptors, PKR1 and PKR2. PKRA83 hydrochloride potently inhibits PK2 receptors with IC50 values of 5.0 nM and 8.2 nM for PKR1 and PKR2, respectively. PKRA83 hydrochloride exhibits anticancer, antiarthritis, and antiangiogenic activities[1].
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Molecular Formula
C27H35Cl2FN2O4
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Molecular Weight
541.48
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Smiles
ClC1=C2C(OCCCO2)=CC(CN(CC(C)C)C([C@H]3CN(CC3)CC4=CC(OC)=C(C=C4)F)=O)=C1.Cl
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Target
Prokineticin Receptor
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Shipping Conditions
Room temperature
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PKRA83 (hydrochloride)
PKRA83 (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.