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Prucalopride (hydrochloride) [CAS 179474-80-7]

Prucalopride (hydrochloride) [CAS 179474-80-7]

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SKU:QM-0064833

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  • Description

    Prucalopride hydrochloride is an orally active, selective and specific 5-HT4 receptor agonist (high affinity), with pKis of 8.6 and 8.1 for human 5-HT4a/4b receptors, respectively. Prucalopride hydrochloride improves intestinal motility by promoting regeneration of the intestinal nervous system in rats. Prucalopride hydrochloride also shows anticancer activity by blocking of the PI3K/AKT/mTor signaling pathway. Prucalopride hydrochloride can be used in studies of chronic constipation, pseudo-intestinal obstruction and cancer[1][2][3].

  • CAS Number

    [179474-80-7]

  • Molecular Formula

    C18H27Cl2N3O3

  • Molecular Weight

    404.33

  • Smiles

    ClC1=C(N)C(CCO2)=C2C(C(NC3CCN(CCCOC)CC3)=O)=C1.Cl

  • Target

    5-HT Receptor

  • Isoform

    5-HT4 Receptor

  • Solubility

    10 mM in DMSO

  • Shipping Conditions

    Room temperature

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Prucalopride (hydrochloride) [CAS 179474-80-7]

Prucalopride (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.