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Pulrodemstat [CAS 1821307-10-1]
Pulrodemstat [CAS 1821307-10-1]
SKU:QM-0061254
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Product Details
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Description
Pulrodemstat (CC-90011) is a potent, selective, reversible and orally active inhibitor of lysine specific demethylase-1 (LSD1) with an IC50 of 0.25 nM. Pulrodemstat is less enzymatic inhibition against LSD2, MOA-A, and MAO-B. Pulrodemstat induces acute myeloid leukemia (AML) and small cell lung cancer (SCLC) cells differentiation and has potent anticancer activity[1].
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CAS Number
[1821307-10-1]
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Molecular Formula
C24H23F2N5O2
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Molecular Weight
451.47
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Smiles
N#CC1=CC=C(C(N=C(N2CCC(N)CC2)N3C)=C(C4=CC=C(OC)C(F)=C4)C3=O)C=C1F
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Target
Histone Demethylase
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Isoform
KDM1/LSD1
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Pulrodemstat [CAS 1821307-10-1]
Pulrodemstat is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.