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Pulrodemstat (Methylbenzenesulfonate) [CAS 2097523-57-2]

Pulrodemstat (Methylbenzenesulfonate) [CAS 2097523-57-2]

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SKU:QM-0061253

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  • Description

    CC-90011 Methylbenzenesulfonate is a potent, selective, reversible and orally active inhibitor of lysine specific demethylase-1 (LSD1) with an IC50 of 0.25 nM. CC-90011 Methylbenzenesulfonate is less enzymatic inhibition against LSD2, MOA-A, and MAO-B. CC-90011 Methylbenzenesulfonate induces acute myeloid leukemia (AML) and small cell lung cancer (SCLC) cells differentiation and has potent anticancer activity[1].

  • CAS Number

    [2097523-57-2]

  • Molecular Formula

    C31H31F2N5O5S

  • Molecular Weight

    623.67

  • Smiles

    N#CC1=CC=C(C(N=C(N2CCC(N)CC2)N3C)=C(C4=CC=C(OC)C(F)=C4)C3=O)C=C1F.O=S(C5=CC=C(C)C=C5)(O)=O

  • Target

    Histone Demethylase

  • Isoform

    KDM1/LSD1

  • Solubility

    10 mM in DMSO

  • Shipping Conditions

    Room temperature

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Pulrodemstat (Methylbenzenesulfonate) [CAS 2097523-57-2]

Pulrodemstat (Methylbenzenesulfonate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.