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Rolapitant (hydrochloride hydrate) [CAS 914462-92-3]

Rolapitant (hydrochloride hydrate) [CAS 914462-92-3]

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QM-0153707-01

£94.75 GBP
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Product Details

  • Description

    Rolapitant hydrochloride hydrate (SCH619734 hydrochloride hydrate) is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a Ki of 0.66 nM. Rolapitant hydrochloride hydrate does not interact with CYP3A4. Rolapitant hydrochloride hydrate shows potent anti-emetic activity in a ferret emesis model[1][2].

  • CAS Number

    [914462-92-3]

  • Molecular Formula

    C25H29ClF6N2O3

  • Molecular Weight

    554.95

  • Smiles

    O=C1N[C@]2(CN[C@@](C3=CC=CC=C3)(CO[C@@H](C4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4)C)CC2)CC1.[H]Cl.O

  • Target

    Neurokinin Receptor

  • Isoform

    NK1R

  • Purity

    98.25

  • Solubility

    DMSO : 250 mg/mL (ultrasonic)

  • Storage Conditions

    4°C (Powder, protect from light)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302

  • Precautions

    H302
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Variant Variant total Quantity Price Variant total
5 mgQM-0153707-01
5 mgQM-0153707-01
£94.75/ea		 £0.00
£94.75/ea £0.00
10 mM - 1 mLQM-0153707-02
10 mM - 1 mLQM-0153707-02
£109.38/ea		 £0.00
£109.38/ea £0.00
10 mgQM-0153707-03
10 mgQM-0153707-03
£136.38/ea		 £0.00
£136.38/ea £0.00
25 mgQM-0153707-04
25 mgQM-0153707-04
£294.22/ea		 £0.00
£294.22/ea £0.00
50 mgQM-0153707-05
50 mgQM-0153707-05
£452.17/ea		 £0.00
£452.17/ea £0.00
100 mgQM-0153707-06
100 mgQM-0153707-06
£702.46/ea		 £0.00
£702.46/ea £0.00
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Rolapitant (hydrochloride hydrate) [CAS 914462-92-3]

Rolapitant (hydrochloride hydrate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.