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SB 243213 (hydrochloride) [CAS 200940-23-4]

SB 243213 (hydrochloride) [CAS 200940-23-4]

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QM-0000228-01

£129.63 GBP
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Product Details

  • Description

    SB 243213 hydrochloride is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 hydrochloride shows greater than a 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels. SB 243213 hydrochloride has improved anxiolytic profile and has the potential for schizophrenia and motor disorders[1].

  • CAS Number

    [200940-23-4]

  • Molecular Formula

    C22H20ClF3N4O2

  • Molecular Weight

    464.87

  • Smiles

    O=C(N1CCC2=C1C=C(C(F)(F)F)C(C)=C2)NC3=CC=C(OC4=CC=CN=C4C)N=C3.[H]Cl

  • Target

    5-HT Receptor

  • Isoform

    5-HT2 Receptor; mLAG-3; MUC2; MUC3; α-1 microglobulin

  • Purity

    98.84

  • Solubility

    10 mM in DMSO

  • Storage Conditions

    4°C (Powder, sealed storage, away from moisture)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302, H312, H332

  • Precautions

    H302, H312, H332
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Variant Variant total Quantity Price Variant total
5 mgQM-0000228-01
5 mgQM-0000228-01
£129.63/ea		 £0.00
£129.63/ea £0.00
10 mgQM-0000228-02
10 mgQM-0000228-02
£238.32/ea		 £0.00
£238.32/ea £0.00
25 mgQM-0000228-03
25 mgQM-0000228-03
£489.83/ea		 £0.00
£489.83/ea £0.00
50 mgQM-0000228-04
50 mgQM-0000228-04
£865.26/ea		 £0.00
£865.26/ea £0.00
100 mgQM-0000228-05
100 mgQM-0000228-05
£1,556.60/ea		 £0.00
£1,556.60/ea £0.00
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SB 243213 (hydrochloride) [CAS 200940-23-4]

SB 243213 (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.