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Talabostat [CAS 149682-77-9]
Talabostat [CAS 149682-77-9]
SKU:QM-0000457-01
£215.24 GBP
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Product Details
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Description
Talabostat (Val-boroPro; PT100) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 Ki = 0.18 nM) and the first clinical inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM), inhibits DPP8/9 (IC50 = 4/11 nM; Ki = 1.5/0.76 nM), quiescent cell proline dipeptidase (QPP) (IC50 = 310 nM), DPP2, and some other DASH family enzymes. Antineoplastic and hematopoiesis- stimulating activities[1][2][3].
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CAS Number
[149682-77-9]
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Molecular Formula
C9H19BN2O3
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Molecular Weight
214.07
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Smiles
CC(C)[C@H](N)C(N1[C@H](B(O)O)CCC1)=O
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Target
Dipeptidyl Peptidase
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Isoform
DPP-4
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Solubility
DMSO : ≥ 40 mg/mL
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Shipping Conditions
Room temperature
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Talabostat [CAS 149682-77-9]
Talabostat is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.