Talabostat (mesylate) [CAS 150080-09-4]
Talabostat (mesylate) [CAS 150080-09-4]
SKU:QM-0143965-01
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Product Details
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Description
Talabostat mesylate (Val-boroPro mesylate; PT100 mesylate) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 Ki = 0.18 nM) and the inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM), inhibits DPP8/9 (IC50 = 4/11 nM; Ki = 1.5/0.76 nM), quiescent cell proline dipeptidase (QPP) (IC50 = 310 nM), DPP2, and some other DASH family enzymes. Antineoplastic and hematopoiesis- stimulating activities[1][2][3].
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CAS Number
[150080-09-4]
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Molecular Formula
C10H23BN2O6S
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Molecular Weight
310.18
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Smiles
CC(C)[C@H](N)C(N1[C@H](B(O)O)CCC1)=O.CS(=O)(O)=O
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Target
Dipeptidyl Peptidase
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Isoform
DPP-4
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Purity
98.35
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Solubility
DMSO : ≥ 40 mg/mL|H2O : 250 mg/mL (ultrasonic)
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Storage Conditions
4°C (Powder, sealed storage, away from moisture)
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Shipping Conditions
Room Temperature
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Hazard Statement
H302, H315, H319, H335
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Precautions
H302, H315, H319, H335
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Talabostat (mesylate) [CAS 150080-09-4]
Talabostat (mesylate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.