Trimegestone-13C, d3
Trimegestone-13C, d3
SKU:QM-0112289
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Product Details
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Description
Trimegestone-13C, d3 is 13C and deuterated labeled Trimegestone. Trimegestone (RU 27987) is an orally active 19-norpregnane progestin. Trimegestone binds to progesterone receptor (PR) with an IC50 value of 3.3 nM (rat PR). Trimegestone increases alkaline phosphatase activity (EC50=0.1 nM) but not luciferase activity. Trimegestone also shows a weak antiandrogenic activity (weak androgen receptor affinity). Trimegestone can be used in studies of contraception or menopausal syndromes[1][2].
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Molecular Formula
C21 13CH27D3O3
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Molecular Weight
346.48
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Smiles
C[C@@]12[C@](CC[C@]2(C)C([C@@H](O)[13C]([2H])([2H])[2H])=O)([H])[C@@]3([H])C(CC1)=C4C(CC3)=CC(CC4)=O
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Target
Androgen Receptor; Isotope-Labeled Compounds; Phosphatase; Progesterone Receptor
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Trimegestone-13C, d3
Trimegestone-13C, d3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.