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TX1-85-1 (Standard) [CAS 1603845-32-4]

TX1-85-1 (Standard) [CAS 1603845-32-4]

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SKU:QM-0002067

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  • Description

    TX1-85-1 (Standard) is the analytical standard of TX1-85-1. This product is intended for research and analytical applications. TX1-85-1 is an irreversible Her3 (ErbB3) inhibitor with an IC50 of 23 nM. TX1-85-1 is also the first selective Her3 ligand, which forms a covalent bond with Cys721 located in the ATP-binding site of Her3. TX1-85-1 induces partial degradation of Her3 protein and attenuates Her3-dependent signaling[1].

  • CAS Number

    [1603845-32-4]

  • Molecular Formula

    C32H36N8O3

  • Molecular Weight

    580.68

  • Smiles

    CC(N1CCN(C2CCC(N3N=C(C4=CC(NC(C=C)=O)=C(OC5=CC=CC=C5)C=C4)C6=C3N=CN=C6N)CC2)CC1)=O

  • Target

    EGFR; Reference Standards

  • Shipping Conditions

    Room temperature

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TX1-85-1 (Standard) [CAS 1603845-32-4]

TX1-85-1 (Standard) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.